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Issue DateTitleAuthor(s)
27-May-2011Jaime E., Charris C.Charris, Jaime
2009Modification of oxidative status in Plasmodium berghei-infected erythrocytes by E-2-chloro-8-methyl-3-[(4’-methoxy-1’-indanoyl)-2’-methyliden]-quinoline compared to chloroquineRodrigues, Juan; Charris, Jaime; Domínguez, José; Ángel, Jorge; Gamboa, Neira
21-Sep-2012N -Formyl-2-(5-nitrothiophen-2-yl)benzothiazole-6-Rodrigues, Juan; Charris, Jaime; Camacho, José; Barazarte, Arthur; Gamboa, Neira; Nitzsche, Bianca; Hopfner, Michael; Lein, Michael; Jung, Klaus; Abramjuk, Claudia
10-May-1999Novel anti-in£ammatory chalcone derivatives inhibit the induction of nitric oxide synthase and cyclooxygenase-2 in mouse peritoneal macrophagesHerencia, Felipe; Ferrandiz, Ma. L; Ubeda, Amalia; Gullén, Isabel; Dominguez, Jose; Charris, Jaime; Lobo, Gricela
Jun-2023Optimization of the synthesis, in silico ADME/ Tox profiling studies, and evaluation of the antimalarial activity of (7-chloroquinolin-4-ylthio) alkylbenzoate derivativesGutiérrez, Joyce E; Fernandez Moreira, Esteban; Acosta, María E; Ramírez, Hegira; Charris, Jaime
9-Nov-2014Potencial Antiepiléptico de Nuevos Derivados de 5-Bencilideno PirimidinasGuevara, Beatriz A; Lobo, Gricela; Rodriguez, Christan; Colman, Trina; Charris, Jaime
1-Oct-2012Potential antitumor and pro-oxidative effects of (E)-methyl 2-(7-chloroquinolin-4-ylthio)-3-(4-hydroxyphenil)acrylate (QNACR)Rodrigues, Juan; Ferrer, Rosa; Gamboa, Neira; Charris, Jaime; Antunes, Fernando
2016Sintesis de 7-cloroquinolinas 4-alquiltiosustituidas. Evaluación de su potencial actividad antimaláricaCharris, Jaime
2006Síntesis y actividad antimalárica de nuevas IsoflavonasDomínguez, José; León, Caritza; Rodrigues, Juan; Gamboa, Neira; Charris, Jaime; Gut, Jiri; Rosenthal, Phillip
23-Aug-2013Síntesis y actividad antimicrobiana de derivados de 4,6-diaminopirimidinas análogos de citosinaLobo, Gricela; Charris, Jaime; Taddei, Antonieta; Monasterios, Melina; Valderrama, Margaret; Romero, Jesús; Charris, Katiuska
23-Aug-2012Síntesis y actividad antimicrobiana de derivados de 4,6-diaminopirimidinas análogos de citosinaLobo, Gricela; Charris, Jaime; Taddei, Antonieta; Monasterios, Melina; Valderrama, Margaret; Romero, Jesis; Charris, Katiuska
2004Stage-specific Activity of Potential Antimalarial Compounds Measured in Vitro by Flow Cytometry in Comparison to Optical Microscopy and Hypoxanthine UptakeCONTRERAS, CARMEN E.; Rivas, María A.; Domínguez, José; Charris, Jaime; Palacios, Mario; Bianco Colmenares, Nicolás E.; Blanca, Isaac
May-2007Synthesis and Antimalarial Activity of Ethyl 3-Amino-4-oxo-9- (phenylsubstituted)thieno[2,3-b]quinoline-2-carboxylate Derivatives.Charris, Jaime; Barazarte, Arthur; Domínguez, José; Lobo, Gricela; Camacho, José; Ferrer, Rosa; Gamboa, Neira; Rodrigues, Juan
6-Dec-2022Synthesis and Antitrypanosomal and Mechanistic Studies of a Series of 2‑Arylquinazolin-4-hydrazines: A Hydrazine Moiety as a Selective, Safe, and Specific Pharmacophore to Design Antitrypanosomal Agents Targeting NO ReleaseRomero, Angel H.; Aguilera, Elena; Gotopo Bastardo, Lourdes Andreina; Charris, Jaime; Rodríguez, Noris; Oviedo, Henry; Dávila, Belén; Cabrera, Gustavo; Cerecetto, Hugo
1-Feb-2011Synthesis and biological evaluation of benzimidazole-5-carbohydrazide derivatives as antimalarial, cytotoxic and antitubercular agentsCamacho, José; Barazarte, Arthur; Gamboa, Neira; Rodrigues, Juan; Rojas, Rosario; Vaisberg, Abraham; Gilman, Robert; Charris, Jaime
15-Apr-2011Synthesis and crystal structure of (4bRS,9bRS)-5-(2,4-dimethoxyphenyl)-4b,9b-7,7-dimethyldihydroxy-4b,5,6,7,8,9b-hexahydroindeno[1,2-b] indole-9,10-dioneLobo, Gricela; Zuleta, Elimar; Charris, Katiuska; Cappareli, Mario; Briceño, Alexander; Ángel, Jorge; Charris, Jaime
18-Apr-2011Synthesis and crystal structure of (4bRS,9bRS)-5-(2,4-dimethoxyphenyl)-4b,9b-7,7-dimethyldihydroxy-4b,5,6,7,8,9b-hexahydroindeno[1,2-b] indole-9,10-dioneLobo, Gricela; Charris, Katiuska; Capparely, Mario; Briceño, Alexander; Ángel, Jorge; Charris, Jaime; Zuleta, Elimar
16-Mar-2020Synthesis and leishmanicidal evaluation of sulfanyl‐and sulfonyl‐tethered functionalized benzoate derivatives featuring a nitroimidazole moietyRodríguez, Miguel; Gutiérrez, Joyce; Domínguez, José; Peixoto, Philippe A.; Fernández, Alexis; Rodríguez, Noris; Deffieux, Denis; Rojas, Luis; Quideau, Stéphane; Pouységu, Laurent; Charris, Jaime
9-Dec-2023Synthesis, Antimalarial, Antileishmanial, and Cytotoxicity Activities and Preliminary In Silico ADMET Studies of 2-(7-Chloroquinolin-4-ylamino)ethyl Benzoate DerivativesGutiérrez, Joyce E.; Ramírez, Hegira; Moreira Fernández, Esteban; Acosta, María E.; Mijares, Michael R.; De Sanctis, Juan Bautista; Gurská, Soňa; Džubák, Petr; Hajdúch, Marián; Labrador Fagúndez, Liesangerli; Stella, Bruno G.; Díaz Pérez, Luis José; Benaim, Gustavo; Charris, Jaime
21-Jul-2023Synthesis of Benzocycloalkanone-Based Michael Acceptors and Biological Activities as Antimalarial and Antitrypanosomal AgentsMijoba, Ali; Fernandez Moreira, Esteban; Parra Giménez, Nereida; Espinosa Tapia, Sandra; Blanco, Zuleyma; Ramírez, Hegira; Charris, Jaime
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